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Drug of the week
An hNK-1 Antagonist
Chien-Yi Chen
Sep 6, 2025
(+)-JRT
Artem Lykov
Jul 18, 2025
AZD5991
Cheng Yang
May 9, 2025
RMC-6291
Emma Simmons
Mar 29, 2025
TRPV3 Antagonist
Chien-Yi Chen
Jan 25, 2025
MK-4256
Yiannakis Lysandrou
Nov 23, 2024
IL-17A Inhibitor Analog 26
Kayla Landers
Sep 28, 2024
Eliquis (BMS)
Eric Pettipiece
Aug 31, 2024
MK-1084
Emma Simmons
Jul 27, 2024
IPI-926 (Saridegib)
Yiannakis Lysandrou
May 4, 2024
AZD8154
Chien-Yi Chen
Mar 23, 2024
Vorolanib (Xcovery)
Bobby Gilbert
Jan 24, 2024
MK-1468
Emma Simmons
Dec 16, 2023
GDC-0022 (Genentech)
Sam Barlock
Nov 11, 2023
PET Imager (1st Biotherapeutics)
David Ryffel
Sep 16, 2023
Zimlovisertib (PF-06650833)
Chris Davis
Jul 29, 2023
Cobimetinib (Genentech)
Zhaochen Duan
Jun 30, 2023
GDC-2394
Yiannakis Lysandrou
Jun 3, 2023
Tavneos (Avacopan)
Jonathan Maturano
Apr 1, 2023
INE963 (Novartis)
David Ryffel
Feb 4, 2023
JDQ443(Novartis)
Chein-Yi Chen
Jan 7, 2023
RGT-068A (Regor Therapeutics Group)
Jingyang Zhang
Nov 19, 2022
Fostemsavir (Rukobia)
Siqi Dong
Oct 8, 2022
Pacritinib (SB1518)
Annie Hooper
Jun 4, 2022
Nitrous Oxide
Chris Davis
Apr 30, 2022
rislenemdaz
Jonathan Maturano
Apr 1, 2022
CoV-2 Therapeutics (Paxlovid)
Peter Ryffel
Jan 22, 2022
molnupiravir
Jonathan Maturano
Oct 8, 2021
Milvexian
David Ryffel
Sep 10, 2021
ARV-471
Annie Hooper
Jul 24, 2021
Ozanimod (Zeposia)
Marko Nesic
Jun 19, 2021
Nirapirib (ZEJULA)
Amanda Milkovits
May 22, 2021
Runcaciguat (BAY 1101042)
Maegen Kincanon
May 1, 2021
Encequidar
David Ryffel
Apr 24, 2021
Tepotinib (Tepmetko)
Annie Hooper
Mar 27, 2021
Lifitegrast (Xiidra)
Marko Nesic
Feb 27, 2021
Phototrexate
Jonathan Maturano
Jan 30, 2021
PF-07059013
David Ryffel
Jan 9, 2021
Pamiparib
David Ryffel
Dec 4, 2020
Orkambi (Lumacaftor and Ivacaftor)
Maegen Kincanon
Nov 13, 2020
Tagrisso (Osimertinib)
Matt Bock
Oct 30, 2020
Fosravuconazole L-lysine ethanolate (Nailin®)
Marko Nesic
Oct 16, 2020
Dextromethorphan
Chris Davis
Sep 25, 2020
Buprenorphine (Subutex) and Naloxone (Narcan)
Christopher J. Huck
Sep 4, 2020
BMS-986260
Tanner Bingham
Aug 21, 2020
Glecaprevir (ABT-493)
Maegen Kincanon
Jul 31, 2020
Maraviroc
Matt Bock
Jul 17, 2020
Temozolomide (TemodarTM)
Marko Nesic
Jul 3, 2020
Selpercatinib (Retevmo ®)
Alexander S. Shved
Jun 5, 2020
Fosfomycin
Christopher J. Huck
May 22, 2020
Alprazolam (Xanax)
Tanner Bingham
May 8, 2020
AMG 510
D. G. Dennis
Apr 24, 2020
GSK2982772
Peter Ryffel
Apr 10, 2020
Spinosyn A (Spinosad)
Jan Petrovcic
Apr 3, 2020
Zepatier (Merck)
Marko Nesic
Mar 27, 2020
Vericiguat (Merck)
Peter Ryffel
Feb 22, 2020
Balovaptan
David Ryffel
Jan 30, 2020
Solifenacin (Vesicare)
Maegen Kincanon
Jan 10, 2020
Coartem®
Daniel Szczepankiewicz
Dec 6, 2019
Imbruvica (Ibrutinib)
Matt Bock
Nov 15, 2019
Palbociclib (Ibrance)
Annie Hooper
Nov 1, 2019
Carmegliptin
Marko Nesic
Oct 4, 2019
Methylphenidate (Ritalin)
Annie Hooper
Sep 20, 2019
Pevonedistat
Daniel Szczepankiewicz
Sep 6, 2019
Larotrectinib (Vitrakvi®)
Matt Bock
Aug 16, 2019
(–)-galantamine
Zohaib Siddiqi
Jul 26, 2019
Lorlatinib
Lucas Hernandez
Apr 19, 2019
Moxifloxacin
Annie Hooper
Feb 15, 2019
Reboxetine (Edronax™)
Daniel Szczepankiewicz
Feb 1, 2019
Salmeterol
Zohaib Siddiqi
Jan 4, 2019
Suvorexant (Belsomra ®)
Bowie Yi
Nov 2, 2018
Emtricitabine (Emtriva ®)
Chad N. Ungarean
Oct 19, 2018
Ketamine
Tanner W. Bingham
Sep 28, 2018
Clopidogrel (Plavix) / Prasugrel (Effient)
Mikiko Okumura
Sep 7, 2018
Cipargamin: Hit Discovery and Drug Development
Yaroslav D. Boyko
Aug 24, 2018
Adventures in Atropisomerism
William C. Wertjes
Aug 10, 2018
Fludeoxyglucose-F18
Alexander S. Shved
Jul 28, 2018
Trabectedin
Emma H. Southgate
Jun 29, 2018
MD-4251 (University of Michigan)
Eric Pettipiece
Aug 16, 2025
Zelquistinel (Syndelio)
Julio Cacho Bravo
Jun 6, 2025
PF-07907063 (Pfizer)
Aaron (Shengshu) Lin
Apr 26, 2025
Deucravacitinib (BMS-986165)
Tsukasa Tawatari
Feb 22, 2025
PF-07265028
Cheng Yang
Dec 14, 2024
ABBV-467
Chien-Yi Chen
Oct 26, 2024
GSK3335103 (GlaxoSmithKline)
Bobby Gilbert
Sep 14, 2024
NX-1607 (Nurix Therapeutics)
Jingyang Zhang
Aug 10, 2024
7-Azaindenoisoquinolines
Zhaochen Duan
Jun 15, 2024
CBPD-268
Cheng Yang
Apr 20, 2024
Suzetrigine (VX-548, Vertex)
Jingyang Zhang
Feb 10, 2024
Aficamten (CK-274)
Eric Pettipiece
Jan 13, 2024
KRAS-G12D Inhibitors
Cheng Yang
Dec 2, 2023
Atogepant (Qulipta™)
Jonathan Maturano
Oct 14, 2023
Loratadine (Claritin)
Chris Davis
Sep 2, 2023
MB076
Jan Petrovcic
Jul 15, 2023
BD-9136
Jingyang Zhang
Jun 17, 2023
PF-06751979 (Pfizer)
Emma Simmons
May 13, 2023
MK-8189
Tsukasa Shimakawa
Feb 25, 2023
Spectinomycin
Chris Davis
Jan 21, 2023
GSK3640254 Derivative
Jan Petrovcic
Dec 10, 2022
A Tetrahydrofluorene Estrogen Receptor Beta Agonist (Merck)
Chris Davis
Oct 15, 2022
GDC-5338 (Genentech)
David Ryffel
Aug 27, 2022
AZD4625
Jingyang Zhang
May 21, 2022
Nonpeptidic HIV‑1 Protease Inhibitors
Matteo Martinelli
Apr 16, 2022
Non-Nucleotide STING Agonists (BMS)
David Ryffel
Feb 26, 2022
Umibecestat
Peter Ryffel
Oct 22, 2021
GSK251
Maegen Kincanon
Sep 24, 2021
Melarsoprol
Chris Davis
Aug 27, 2021
Fosdenopterin (Nulibry)
Zohaib Siddiqi
Jul 3, 2021
Azithromycin (Zithromax)
Roberto Serrano
Jun 5, 2021
Daprodustat
Peter Ryffel
May 8, 2021
Etoposide
Chris Davis
Apr 24, 2021
AZD5718
Tanner Bingham
Apr 10, 2021
Baloxivir Marboxil (Xofluza)
Zohaib Siddiqi
Mar 13, 2021
Fluticasone propionate
Amanda Milkovits
Feb 6, 2021
Koseluga (Selumetinib)
Maegen Kincanon
Jan 16, 2021
Psilocybin
Annie Hooper
Dec 19, 2020
PF-06835919
Tanner Bingham
Nov 20, 2020
Abrocitinib (PF-04965842)
Daniel Szczepankiewicz
Nov 6, 2020
Entecavir (Baraclude®)
Sungjong Lee
Oct 23, 2020
Zepzelca (Lurbinectedin)
D. G. Dennis
Oct 9, 2020
Avapritinib (Ayvakit)
Annie Hooper
Sep 11, 2020
ETX0282
David Ryffel
Aug 28, 2020
Rimegepant
D. G. Dennis
Aug 14, 2020
Sacituzumab Govitecan-hziy (Trodelvy™)
Daniel Szczepankiewicz
Jul 24, 2020
Bictegravir (Biktarvy®)
Sungjong Lee
Jul 10, 2020
Clindamycin
Chris Davis
Jun 12, 2020
Carfilzomib
Annie Hooper
May 29, 2020
Remdesivir (GS-5734)
David Ryffel
May 15, 2020
Bryostatin 1
Roberto Serrano
May 1, 2020
Ubrelvy (Ubrogepant)
Maegen Kincanon
Apr 17, 2020
LOU064 (Remibrutinib)
Matt Bock
Apr 3, 2020
amlodipine
Zohaib Siddiqi
Mar 27, 2020
Taniborbactam (VNRX-5133)
Sungjong Lee
Mar 5, 2020
Tropifexor (LJN452)
Sungjong Lee
Feb 6, 2020
[𝛹[C(=NH)NH]Tpg⁴]vancomycin and Related Analogues
Christopher J. Huck
Jan 24, 2020
Verubecestat (MK-8931)
Daniel Szczepankiewicz
Dec 20, 2019
MK-8719
Chad N. Ungarean
Nov 22, 2019
Sofosbuvir (PSI-7977)
Sungjong Lee
Nov 8, 2019
Rolapitant (Varubi™)
Marko Nesic
Oct 11, 2019
Eravacycline (XeravaTM)
David G. Dennis
Sep 27, 2019
Tectin®
Yaroslav D. Boyko
Sep 13, 2019
Lubiprostone
Zohaib Siddiqi
Aug 23, 2019
Aprepitant (Emend™)
Daniel Szczepankiewicz
Aug 2, 2019
AZD6738
Sungjong Lee
Jul 19, 2019
Saxagliptin
Marko Nesic
Mar 15, 2019
The Antifungal Pipeline: Voriconazole and beyond
Yaroslav D. Boyko
Feb 8, 2019
Rivaroxaban (Xarelto ®)
Matt Bock
Jan 18, 2019
Bicyclic Iminopyrimidinone BACE1 Inhibitors
Lucas W. Hernandez
Nov 30, 2018
Escitalopram
William C. Wertjes
Oct 26, 2018
Fentanyl
Emma H. Southgate
Oct 5, 2018
Lusutrombopag (Mulpleta ®)
Alexander S. Shved
Sep 21, 2018
Linezolid (Zyvox ®)
Bowie Yi
Aug 31, 2018
Ambien® (Zolpidem Tartrate)
David G. Dennis
Aug 17, 2018
Rucaparib Camsylate (Rubraca)
Conghui Tang
Aug 2, 2018
Risperidone
Emma H. Southgate
Jul 20, 2018
Dolutegravir
Bowie Yi
Jun 29, 2018
Archive
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